SCHEMBL4731297

SCHEMBL4731297

COC(=O)c1sc(-c2ccc(-c3cc4ncccn4n3)cc2)cc1N(C(=O)c1ccc(C(F)(F)F)cc1C(F)(F)F)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 1/20 0.33
GFER P55789 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 4/20 0.33
CYP2B6 P20813 4/20 0.33
CYP2C19 P33261 3/20 0.33
CYP3A4 P08684 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C8 P10632 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 2/20 0.32
IKBKB O14920 1/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731374 0.94 NTRK1 (0.34) NPSR1MAPTKDM4EMAPK1GFER
SCHEMBL4731314 0.93 APOBEC3A (0.33) ALDH1A1CYP2C9CYP2B6CYP2C19CYP3A4
SCHEMBL4732780 0.86 NTRK1 (0.34) ALDH1A1
SCHEMBL4731338 0.86 IRAK4 (0.35) MAPT
SCHEMBL4730446 0.85 KDM4E (0.38) TP53RXFP1NPSR1MAPTKDM4E
SCHEMBL4727903 0.84 MAPT (0.39) TP53RXFP1NPSR1MAPTKDM4E
SCHEMBL4732282 0.84 KDM4E (0.32) NPSR1MAPTKDM4EALDH1A1CYP2C9
SCHEMBL4139806 0.80 KDM4E (0.36) KDM4EHPGDIKBKB
SCHEMBL4139800 0.80 KDM4E (0.36) KDM4EHPGDIKBKB
SCHEMBL4798458 0.78 APOBEC3A (0.33) CYP2C9CYP2B6CYP2C19CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed