SCHEMBL4730446

SCHEMBL4730446

COC(=O)c1sc(-c2ccc(-c3cc4ncccn4n3)cc2)cc1N(C(=O)c1ccc(Cl)cc1F)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
NPSR1 Q6W5P4 2/20 0.36
IKBKB O14920 1/20 0.34
RXFP1 Q9HBX9 2/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 2/20 0.34
POLB P06746 2/20 0.32
TGFBR1 P36897 1/20 0.32
MCOLN3 Q8TDD5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4727903 0.93 MAPT (0.39) KDM4EMAPTNPC1CASP3RAB9A
SCHEMBL4730991 0.93 APOBEC3A (0.33) KDM4ENPC1RAB9ATP53
SCHEMBL4731374 0.90 NTRK1 (0.34) KDM4EMAPTNPSR1IKBKBPOLB
SCHEMBL4731338 0.86 IRAK4 (0.35) MAPT
SCHEMBL4728477 0.86 SLC6A9 (0.35) RXFP1TP53
SCHEMBL14223294 0.86 NPC1 (0.37) KDM4EMAPTNPC1CASP3RAB9A
SCHEMBL14223017 0.85 KDM4E (0.33) KDM4EMAPTNPC1CASP3RAB9A
SCHEMBL4732282 0.85 KDM4E (0.32) KDM4EMAPTNPC1CASP3RAB9A
SCHEMBL4732771 0.85 APOBEC3A (0.34) KDM4ENPC1RAB9ATP53
SCHEMBL4731297 0.85 TP53 (0.34) KDM4EMAPTNPSR1IKBKBRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed