SCHEMBL4732072

SCHEMBL4732072

NC(=O)[C@H]1CCc2cccc(-c3c(Cl)cccc3Cl)c2O1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NFKB1 P19838 6/20 0.39
NFKB2 Q00653 6/20 0.39
RELA Q04206 6/20 0.39
FABP4 P15090 7/20 0.38
FABP3 P05413 1/20 0.38
PARP1 P09874 1/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
AQP1 P29972 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731714 1.00 TDP1 (0.40) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL8213736 0.89 SMN1; SMN2 (0.41) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL4729890 0.89 SMN1; SMN2 (0.41) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL8203895 0.89 SMN1; SMN2 (0.41) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL4732206 0.85 L3MBTL1 (0.42) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL8209908 0.77 TDP1 (0.34) TDP1L3MBTL1FABP4FABP3AQP1
SCHEMBL8258102 0.77 AQP1 (0.42) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL8255634 0.77 AQP1 (0.42) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL4621299 0.77 AQP1 (0.42) TDP1L3MBTL1NFKB1NFKB2RELA
SCHEMBL5324235 0.76 TDP1 (0.39) TDP1L3MBTL1FABP4FABP3AQP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052087-A1 CHROMANE DERIVATIVES AND USES THEREOF WYETH (US) 2008-05-02 WO disclosed
WO-2008052088-A1 CHROMANE DERIVATIVES, SYNTHESIS THEREOF, AND INTERMEDIATES THERETO WYETH (US) 2008-05-02 WO disclosed
WO-2008052088-A1 CHROMANE DERIVATIVES, SYNTHESIS THEREOF, AND INTERMEDIATES THERETO WYETH (US) 2008-05-02 WO disclosed