SCHEMBL4732088

SCHEMBL4732088

COc1ccncc1C=CC(=O)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP17A1 P05093 8/20 0.43
CYP19A1 P11511 8/20 0.43
CYP1A1 P04798 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1B1 Q16678 2/20 0.42
CYP3A4 P08684 1/20 0.42
TOP2A P11388 1/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8216865 0.85 RAB9A (0.36) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL5510876 0.79 JUN (0.60) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL4729644 0.76 CNR2 (0.46) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL8068014 0.74 JUN (0.51) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL6092331 0.74 JUN (0.51) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL8077622 0.73 MAPT (0.56) MEN1KMT2AMAPTCYP17A1CYP19A1
SCHEMBL1769996 0.73 MAPT (0.56) MEN1KMT2AMAPTCYP17A1CYP19A1
SCHEMBL16052805 0.72 ALDH1A1 (0.56) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL5509239 0.72 ALDH1A1 (0.56) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL4728511 0.72 ALDH1A1 (0.61) MEN1KMT2AALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed