SCHEMBL4730918

SCHEMBL4730918

CC1(C)c2cc(OC(F)(F)F)ccc2S(=O)(=O)c2cc(F)ccc21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 4/20 0.39
VEGFA P15692 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.33
CES1 P23141 1/20 0.33
ABL1 P00519 1/20 0.31
TRPV4 Q9HBA0 2/20 0.31
SLC40A1 Q9NP59 1/20 0.31
CTSL P07711 1/20 0.31
GALR1 P47211 1/20 0.30
SCN8A Q9UQD0 1/20 0.30
SCN10A Q9Y5Y9 1/20 0.30
HSPA9 P38646 1/20 0.30
KIF11 P52732 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730920 0.85 GPR3 (0.39) GPR3VEGFAPTGDR2TRPV4SCN8A
SCHEMBL4732090 0.75 AGBL2 (0.34)
SCHEMBL4733537 0.74 GPR3 (0.40) GPR3CES1ABL1TRPV4SLC40A1
SCHEMBL4730728 0.73 BACE1 (0.35)
SCHEMBL4733059 0.67 TRPV4 (0.33) TRPV4
SCHEMBL4782389 0.66 ATM (0.41)
SCHEMBL4734722 0.64 HCAR3 (0.33)
SCHEMBL4733543 0.63 GPR3 (0.40) GPR3PTGDR2CES1TRPV4CTSL
SCHEMBL31536406 0.62 BACE1 (0.37) CES1SLC40A1CTSLHSPA9
SCHEMBL2264074 0.62 CES1 (0.51) CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed