SCHEMBL4735360

SCHEMBL4735360

CCOC(=O)[C@H](Cc1ccc(Nc2ncccc2[N+](=O)[O-])cc1)NC(=O)c1c(Cl)cncc1Cl

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 13/20 0.62
ITGB1 P05556 13/20 0.62
MAPT P10636 2/20 0.55
NPC1 O15118 1/20 0.55
NFKB1 P19838 1/20 0.55
MAPK1 P28482 1/20 0.55
RAB9A P51151 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55
CYP3A4 P08684 1/20 0.40
ALDH1A1 P00352 3/20 0.40
ITGB3 P05106 1/20 0.40
ITGAV P06756 1/20 0.40
ITGA5 P08648 1/20 0.40
ITGA2 P17301 1/20 0.38
ITGB7 P26010 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736051 0.91 ITGB1 (0.54) ITGA4ITGB1MAPTNPC1NFKB1
SCHEMBL4734982 0.86 ITGA4 (0.49) ITGA4ITGB1CYP3A4ITGB3ITGAV
SCHEMBL4734738 0.81 MAPT (0.59) ITGA4ITGB1MAPTNPC1NFKB1
SCHEMBL4730913 0.79 MAPT (0.67) ITGA4ITGB1MAPTNPC1NFKB1
SCHEMBL4735069 0.78 ITGB1 (0.41) ITGA4ITGB1CYP3A4ITGB3ITGAV
SCHEMBL5374019 0.77 ITGB1 (1.00) ITGA4ITGB1
SCHEMBL4736909 0.76 MAPT (0.56) ITGA4ITGB1MAPTNPC1NFKB1
SCHEMBL1414434 0.75 MAPT (0.70) ITGA4ITGB1MAPTNPC1NFKB1
SCHEMBL4733784 0.73 MAPT (0.52) ITGA4ITGB1MAPTNPC1NFKB1
SCHEMBL4733947 0.73 MAPT (0.52) MAPTNPC1NFKB1MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed