SCHEMBL4736051

SCHEMBL4736051

CCOC(=O)[C@H](Cc1cccc(Nc2ncccc2[N+](=O)[O-])c1)NC(=O)c1c(Cl)cncc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 8/20 0.54
ITGA4 P13612 6/20 0.54
MAPT P10636 4/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
MAPK1 P28482 2/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
ALDH1A1 P00352 5/20 0.39
JAK2 O60674 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
CYP3A4 P08684 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
ITGB7 P26010 1/20 0.37
ITGA5 P08648 3/20 0.37
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4735360 0.91 ITGA4 (0.62) ITGB1ITGA4MAPTNPC1RAB9A
SCHEMBL4735069 0.87 ITGB1 (0.41) ITGB1ITGA4CYP3A4ITGB7ITGA5
SCHEMBL4733947 0.82 MAPT (0.52) MAPTNPC1RAB9AMAPK1NFKB1
SCHEMBL4733395 0.80 MAPT (0.58) MAPTNPC1RAB9AMAPK1NFKB1
SCHEMBL4734982 0.78 ITGA4 (0.49) ITGB1ITGA4CYP3A4ITGB7ITGA5
SCHEMBL4734738 0.73 MAPT (0.59) ITGB1ITGA4MAPTNPC1RAB9A
SCHEMBL6797565 0.72 MAPT (0.78) MAPTNPC1RAB9AMAPK1NFKB1
SCHEMBL6797448 0.71 LMNA (0.55) MAPTNPC1RAB9AMAPK1NFKB1
SCHEMBL5374019 0.70 ITGB1 (1.00) ITGB1ITGA4
SCHEMBL1414433 0.70 MAPT (0.62) ITGB1ITGA4MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed