SCHEMBL4735544

SCHEMBL4735544

CCN(C(=O)c1c(Cl)cncc1Cl)[C@@H](Cc1ccc(-n2c([C@@H]3CCCCN3)nc3cccnc32)cc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 17/20 0.53
ITGA4 P13612 17/20 0.53
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PDE4B Q07343 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736084 0.83 ITGA4 (0.62) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL4736103 0.83 ITGA4 (0.62) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL4732547 0.83 ITGA4 (0.62) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL4734892 0.82 SIGMAR1 (0.39) ITGB1ITGA4
SCHEMBL4733969 0.80 ITGA4 (0.54) ITGB1ITGA4MEN1KMT2APDE4B
SCHEMBL4730854 0.77 ITGB1 (0.64) ITGB1ITGA4
SCHEMBL4730816 0.77 ITGB1 (0.64) ITGB1ITGA4
SCHEMBL4735182 0.74 ITGB1 (0.55) ITGB1ITGA4MEN1KMT2APDE4B
SCHEMBL4735900 0.72 ITGB1 (0.70) ITGB1ITGA4CYP3A4CYP2C9
SCHEMBL4737683 0.72 ITGB1 (0.70) ITGB1ITGA4CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed