SCHEMBL4735546

SCHEMBL4735546

C#CC1CCCCC1NC(=O)c1cccnc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 3/20 0.44
TAS1R1 Q7RTX1 3/20 0.44
TAS1R2 Q8TE23 3/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HCRTR1 O43613 2/20 0.43
CHRM1 P11229 2/20 0.43
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RAB9A P51151 2/20 0.42
MAPT P10636 1/20 0.42
NPC1 O15118 1/20 0.41
ACKR3 P25106 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9155166 0.81 TAS1R3 (0.63) TAS1R3TAS1R1TAS1R2ALDH1A1KDM4E
SCHEMBL22449342 0.81 GRM5 (0.56) ALDH1A1GAAKDM4ESMN1; SMN2RAB9A
SCHEMBL26655975 0.78 ALDH1A1 (0.49) TAS1R3TAS1R1TAS1R2ALDH1A1GAA
SCHEMBL9153874 0.78 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2ALDH1A1GAA
SCHEMBL9157091 0.78 HSD11B1 (0.48) TAS1R3TAS1R1TAS1R2ALDH1A1GAA
SCHEMBL3165964 0.78 ALDH1A1 (0.68) ALDH1A1GAAKDM4ELMNASMN1; SMN2
SCHEMBL4736777 0.77 SIGMAR1 (0.43) TAS1R3TAS1R1TAS1R2ALDH1A1GAA
SCHEMBL31583752 0.76 P2RX7 (0.58) ALDH1A1GAAKDM4ELMNASMN1; SMN2
SCHEMBL6063992 0.72 P2RX7 (0.54) ALDH1A1GAAKDM4ELMNASMN1; SMN2
SCHEMBL27894457 0.71 SMN1; SMN2 (0.56) ALDH1A1GAAKDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008081017-A1 NEW N-ALKYNYLCARBOXAMIDE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2008-07-10 WO disclosed