SCHEMBL4735753

SCHEMBL4735753

CCOC(=O)C1=C(C(F)(F)F)C2C=C(C)C1O2

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
KDM4E B2RXH2 5/20 0.37
ADORA2B P29275 2/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
IDO1 P14902 1/20 0.35
LMNA P02545 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
GAA P10253 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ABCC1 P33527 1/20 0.33
ATM Q13315 1/20 0.33
TP53 P04637 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
CACNA1C Q13936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4735732 0.89 HDAC4 (0.38) HDAC4HDAC6KDM4EADORA2BHDAC3
SCHEMBL4739182 0.78 HDAC4 (0.41) HDAC4HDAC6KDM4EADORA2BHDAC3
SCHEMBL12286063 0.69 HDAC4 (0.41) HDAC4HDAC6KDM4EADORA2BHDAC3
SCHEMBL18501088 0.66 HDAC4 (0.38) HDAC4HDAC6KDM4EADORA2BHDAC3
SCHEMBL31376339 0.66 KDM4E (0.46) KDM4ELMNAALDH1A1TSHRGAA
SCHEMBL19543293 0.62 KDM4E (0.42) HDAC4HDAC6KDM4ELMNAALDH1A1
SCHEMBL9726284 0.61 KDM4E (0.62) KDM4EADORA2BLMNAALDH1A1TSHR
SCHEMBL19543295 0.61 ADORA3 (0.47) KDM4ELMNAALDH1A1TSHRGAA
SCHEMBL9225568 0.60 HDAC4 (0.38) HDAC4HDAC6KDM4EADORA2BHDAC3
SCHEMBL6731339 0.60 KDM4E (0.64) KDM4EIDO1LMNAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075955-A2 PROCESS FOR THE PREPARATION OF 1,4,5-TRISUBSTITUTED TRIAZOLES AND 3,4,5-TRISUBSTITUTED TRIAZOLES STICHTING VOOR DE TECHNISCHE WETENSCHAPPEN (NL) 2008-06-26 WO disclosed
WO-2008075955-A2 PROCESS FOR THE PREPARATION OF 1,4,5-TRISUBSTITUTED TRIAZOLES AND 3,4,5-TRISUBSTITUTED TRIAZOLES STICHTING VOOR DE TECHNISCHE WETENSCHAPPEN (NL) 2008-06-26 WO disclosed