SCHEMBL4736673

SCHEMBL4736673

O=C(CC1CCCN(S(=O)(=O)c2ccccc2F)C1)NN1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
EPHX2 P34913 1/20 0.49
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
LMNA P02545 4/20 0.46
CNR2 P34972 1/20 0.45
CHRNB2 P17787 2/20 0.45
CHRNB4 P30926 2/20 0.45
CHRNA3 P32297 2/20 0.45
CHRNA4 P43681 2/20 0.45
CYP19A1 P11511 1/20 0.43
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4808038 0.91 MAPT (0.48) ALDH1A1EPHX2CYP3A4CYP2C19LMNA
SCHEMBL4741684 0.90 ALDH1A1 (0.49) ALDH1A1EPHX2CYP3A4CYP2C19LMNA
SCHEMBL4785880 0.89 CYP3A4 (0.46) CYP3A4CYP2C19LMNAPKMSMN1; SMN2
SCHEMBL4736649 0.87 CYP3A4 (0.50) ALDH1A1EPHX2CYP3A4CYP2C19LMNA
SCHEMBL4740746 0.87 CYP3A4 (0.50) ALDH1A1EPHX2CYP3A4CYP2C19LMNA
SCHEMBL4737578 0.87 EPHX2 (0.49) ALDH1A1EPHX2CYP2C19LMNACNR2
SCHEMBL4739746 0.87 HDAC3 (0.52) CYP3A4CYP2C19LMNASMN1; SMN2
SCHEMBL4740922 0.87 CYP19A1 (0.43) ALDH1A1CYP3A4CYP2C19LMNACYP19A1
SCHEMBL4738916 0.87 HDAC3 (0.52) CYP3A4CYP2C19LMNASMN1; SMN2
SCHEMBL4736709 0.86 LMNA (0.57) ALDH1A1CYP3A4CYP2C19LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO claimed
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO disclosed