SCHEMBL4736736

SCHEMBL4736736

NC(=O)C1CCCN(c2ccc(CN(C(=O)c3cccnc3)c3ccc(F)cc3)cn2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.44
TSHR P16473 2/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 3/20 0.42
VNN1 O95497 1/20 0.41
FPR2 P25090 1/20 0.40
SCN9A Q15858 1/20 0.40
ALDH1A1 P00352 2/20 0.39
OPRM1 P35372 2/20 0.39
OPRK1 P41145 1/20 0.39
PDK1 Q15118 2/20 0.39
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
OPRD1 P41143 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAPK14 Q16539 1/20 0.37
CXCR2 P25025 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736742 0.90 GAA (0.46) TSHRGAAKMT2AVNN1OPRM1
SCHEMBL4787168 0.89 TSHR (0.45) TSHRGAAKMT2AVNN1ALDH1A1
SCHEMBL4738973 0.88 TSHR (0.44) TSHRGAAKMT2AVNN1FPR2
SCHEMBL4735150 0.86 TSHR (0.51) TSHRGAAKMT2AALDH1A1OPRM1
SCHEMBL4786168 0.86 TSHR (0.47) TSHRGAAVNN1ALDH1A1OPRM1
SCHEMBL4737958 0.84 TSHR (0.48) TSHRGAAVNN1ALDH1A1OPRM1
SCHEMBL4735235 0.82 GAA (0.47) TSHRGAAOPRM1PDK1KDM4E
SCHEMBL4733572 0.82 TSHR (0.45) TSHRGAAALDH1A1OPRM1OPRK1
SCHEMBL4736729 0.82 TSHR (0.46) TSHRGAAALDH1A1OPRM1OPRK1
SCHEMBL4738239 0.81 TSHR (0.49) TSHRGAAALDH1A1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed