SCHEMBL4738973

SCHEMBL4738973

O=C(c1cccnc1)N(Cc1ccc(N2CCCC(CO)C2)nc1)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
GAA P10253 1/20 0.44
PDK1 Q15118 2/20 0.39
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
MAPK14 Q16539 1/20 0.37
CXCR2 P25025 1/20 0.37
KMT2A Q03164 1/20 0.37
RORC P51449 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
FPR1 P21462 1/20 0.36
FPR2 P25090 1/20 0.36
VNN1 O95497 1/20 0.36
HTT P42858 1/20 0.36
SMO Q99835 1/20 0.36
HSD17B10 Q99714 1/20 0.36
FAAH O00519 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787168 0.90 TSHR (0.45) TSHRGAAPDK1MAPK14CXCR2
SCHEMBL4735235 0.90 GAA (0.47) TSHRGAAPDK1MAPK14CXCR2
SCHEMBL4736736 0.88 CDK9 (0.44) TSHRGAAPDK1MAPK14CXCR2
SCHEMBL4735150 0.87 TSHR (0.51) TSHRGAAPDK1MAPK14CXCR2
SCHEMBL4786168 0.86 TSHR (0.47) TSHRGAAPDK1KLKB1KLK1
SCHEMBL4738289 0.85 GAA (0.45) TSHRGAAPDK1MAPK14CXCR2
SCHEMBL4737958 0.85 TSHR (0.48) TSHRGAAPDK1MAPK14CXCR2
SCHEMBL3059465 0.84 ACHE (0.40) TSHRKMT2AKDM4EALDH1A1FPR1
SCHEMBL4735626 0.83 TSHR (0.42) TSHRGAAPDK1MAPK14KDM4E
SCHEMBL4733572 0.83 TSHR (0.45) TSHRGAAPDK1MAPK14CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed