SCHEMBL4787168

SCHEMBL4787168

O=C(c1cccnc1)N(Cc1ccc(N2CCCC(O)C2)nc1)c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
GAA P10253 1/20 0.45
PDK1 Q15118 2/20 0.41
CXCR2 P25025 1/20 0.40
VNN1 O95497 1/20 0.40
OPRM1 P35372 2/20 0.39
OPRK1 P41145 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPK14 Q16539 2/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HTT P42858 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SMO Q99835 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
OPRD1 P41143 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786168 0.95 TSHR (0.47) TSHRGAAPDK1CXCR2VNN1
SCHEMBL4738973 0.90 TSHR (0.44) TSHRGAAPDK1CXCR2VNN1
SCHEMBL4737958 0.90 TSHR (0.48) TSHRGAAPDK1CXCR2VNN1
SCHEMBL4736736 0.89 CDK9 (0.44) TSHRGAAPDK1CXCR2VNN1
SCHEMBL4735150 0.89 TSHR (0.51) TSHRGAAPDK1CXCR2OPRM1
SCHEMBL4735235 0.84 GAA (0.47) TSHRGAAPDK1CXCR2OPRM1
SCHEMBL4733572 0.84 TSHR (0.45) TSHRGAAPDK1CXCR2OPRM1
SCHEMBL3064212 0.84 OPRM1 (0.41) TSHROPRM1OPRK1HSD17B10KMT2A
SCHEMBL4736729 0.84 TSHR (0.46) TSHRGAAPDK1CXCR2OPRM1
SCHEMBL4736742 0.84 GAA (0.46) TSHRGAAPDK1CXCR2VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed