SCHEMBL473877

SCHEMBL473877

Cc1cc(Cl)nc(Cl)c1C(=O)O

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.74
MAPK1 P28482 1/20 0.74
SMN1; SMN2 Q16637 1/20 0.74
TAAR1 Q96RJ0 1/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
POLB P06746 1/20 0.50
CYP3A4 P08684 4/20 0.45
ACHE P22303 1/20 0.45
GPR35 Q9HC97 1/20 0.42
DAO P14920 1/20 0.39
MAPT P10636 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
CYP2C19 P33261 2/20 0.38
DHODH Q02127 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HIF1A Q16665 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C8 P10632 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29384281 1.00 ALDH1A1 (0.74) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL2132960 0.88 ALDH1A1 (0.63) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
Hydrochloric Acid SCHEMBL3758009 0.86 ALDH1A1 (0.61) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL11385463 0.86 ALDH1A1 (0.61) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL29434700 0.85 ALDH1A1 (0.55) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL3752932 0.85 ALDH1A1 (0.55) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL3340047 0.85 SMN1; SMN2 (1.00) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL29898229 0.85 SMN1; SMN2 (1.00) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL25282673 0.84 ALDH1A1 (0.59) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1
SCHEMBL8686340 0.84 SMN1; SMN2 (0.80) ALDH1A1MAPK1SMN1; SMN2TAAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 231 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313981-B1 3,4-DIHYDRO-2,7-NAPHTHYRIDINE-1,6(2H,7H)-DIONES AS MEK INHIBITORS PFIZER (US) 2026-02-25 EP disclosed
EP-4676922-A1 BIFUNCTIONAL COMPOUNDS CAPABLE OF DEGRADING ANDROGEN RECEPTORS Astrazeneca AB (SE) 2026-01-14 EP disclosed
EP-3768260-B1 OXADIAZOLE COMPOUNDS AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS HOFFMANN LA ROCHE (CH) 2025-10-08 EP disclosed
EP-4619397-A1 SALT-INDUCIBLE KINASES (SIK) INHIBITORS AND METHODS OF USES THEREOF Insilico Medicine IP Limited (HK) 2025-09-24 EP disclosed
EP-3952870-B1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS NANJING ZENSHINE PHARMACEUTICALS CO LTD (CN) 2025-09-24 EP disclosed
US-20250263411-A1 3,4-DIHYDRO-2,7-NAPHTHYRIDINE-1,6(2H,7H)-DIONES AS MEK INHIBITORS PFIZER INC. (US) 2025-08-21 US disclosed
WO-2025134150-A1 BIPHENYL PYRIDINE RIGID COMPOUNDS WITH POLYCYCLIC HETEROCYCLES USEFUL AS DUAL IMMUNE CHECKPOINT INHIBITORS NATCO PHARMA LIMITED (IN) 2025-06-26 WO disclosed
US-20250177539-A1 ER DEGRADERS AND USES THEREOF ASTRAZENECA AB (SE) 2025-06-05 US disclosed
US-20250154109-A1 SODIUM CHANNEL BLOCKING COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC 2025-05-15 US disclosed
US-20250122184-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2025-04-17 US disclosed
US-20040209866-A1 1,8 Naphthyridine derivatives and their use to treat diabetes and related disorders BAYER PHARMACEUTICALS CORPORATION 2004-10-21 US disclosed
WO-2004083207-A1 NAPHTHYRIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS ABBOTT LABORATORIES (US) 2004-09-30 WO disclosed
US-20040157875-A1 1, 6-Naphthyridine derivatives and their use to treat diabetes and related disorders BAYER PHARMACEUTICALS CORPORATION 2004-08-12 US disclosed
EP-1432710-A1 1, 8-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS Bayer Pharmaceuticals Corporation (US) 2004-06-30 EP disclosed
EP-1432711-A1 1,6-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS Bayer Corporation (US) 2004-06-30 EP disclosed
US-20040014751-A1 1,8-Naphthyridine derivatives and their use to treat diabetes and related disorders BAYER CORPORATION 2004-01-22 US disclosed
US-6677352-B1 1,6-naphthyridine derivatives and their use to treat diabetes and related disorders BAYER PHARMACEUTICALS CORPORATION 2004-01-13 US disclosed
US-20030232818-A1 Antibacterial compounds ABBVIE INC. 2003-12-18 US disclosed
WO-2003027112-A1 1, 8-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed
WO-2003027113-A1 1,6-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250154109-A1 SODIUM CHANNEL BLOCKING COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE SCN8A, TRPV1, SCNN1A ALDH1A1 2842/4885MAPK1 2312/4885SMN1; SMN2 741/4885
US-20040157875-A1 1, 6-Naphthyridine derivatives and their use to treat diabetes and related disorders GLP1R, NQO1, UQCRC1 ALDH1A1 850/4885MAPK1 894/4885SMN1; SMN2 2827/4885
US-20040209866-A1 1,8 Naphthyridine derivatives and their use to treat diabetes and related disorders SLC5A1, NQO1, GLP1R ALDH1A1 754/4885MAPK1 954/4885SMN1; SMN2 2937/4885
US-20040014751-A1 1,8-Naphthyridine derivatives and their use to treat diabetes and related disorders UQCRC1, GLP1R, SLC5A1 ALDH1A1 820/4885MAPK1 1071/4885SMN1; SMN2 3159/4885
US-20030232818-A1 Antibacterial compounds PGLS, UGT1A1, CASP1 ALDH1A1 292/4885MAPK1 341/4885SMN1; SMN2 2135/4885
US-20250263411-A1 3,4-DIHYDRO-2,7-NAPHTHYRIDINE-1,6(2H,7H)-DIONES AS MEK INHIBITORS NRAS, KRAS, BRAF ALDH1A1 1249/4885MAPK1 15/4885SMN1; SMN2 2423/4885
US-20250122184-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS TRPA1, TRPV1, TRPV3 ALDH1A1 721/4885MAPK1 1686/4885SMN1; SMN2 1161/4885
US-20250177539-A1 ER DEGRADERS AND USES THEREOF ESR1, ESR2, ESRRA ALDH1A1 1672/4885MAPK1 2785/4885SMN1; SMN2 455/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.