SCHEMBL473882

SCHEMBL473882

COc1ccc(CBr)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.46
HTR2A P28223 5/20 0.46
KCNH2 Q12809 3/20 0.46
HTR1A P08908 1/20 0.43
APLNR P35414 1/20 0.43
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.40
GFER P55789 1/20 0.40
KDM4E B2RXH2 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29976707 1.00 SLC6A4 (0.46) SLC6A4HTR2AKCNH2HTR1AAPLNR
SCHEMBL474102 0.84 HTR2A (0.46) SLC6A4HTR2AKCNH2HTR1AMEN1
SCHEMBL11530709 0.82 RELA (0.48) MEN1KMT2AALDH1A1KDM4E
SCHEMBL11530716 0.82 RELA (0.48) MEN1KMT2AALDH1A1KDM4E
SCHEMBL4519124 0.82 KDM4E (0.37) SLC6A4HTR2AKCNH2HTR1AMEN1
SCHEMBL4510419 0.82 ALDH1A1 (0.53) SLC6A4HTR2AKCNH2HTR1AAPLNR
SCHEMBL8340513 0.82 SLC6A4 (0.47) SLC6A4HTR2AKCNH2HTR1AAPLNR
SCHEMBL2060421 0.81 HTR2A (0.47) HTR2AAPLNRCA12CA1CA2
SCHEMBL1391304 0.81 NQO1 (0.46) MEN1KMT2AALDH1A1KDM4E
SCHEMBL3719649 0.81 EPHX2 (0.42) SLC6A4HTR2AHTR1AKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 123 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS SHANGHAI SHOUTI BIOTECHNOLOGY CO., LTD. (CN) 2025-04-03 US disclosed
US-11725000-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2023-08-15 US disclosed
CN-110023292-B Apoptosis inhibitors 北京生命科学研究所 2022-10-04 CN disclosed
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
US-20210309647-A1 Apoptosis Inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-10-07 US disclosed
US-11034680-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-06-15 US disclosed
EP-3484854-B1 APOPTOSIS INHIBITORS NAT INSTITUTE OF BIOLOGICAL SCIENCES BEIJING (CN) 2021-01-20 EP disclosed
EP-2432776-B1 METHYL SULFANYL PYRIMIDINES USEFUL AS ANTIINFLAMMATORIES, ANALGESICS, AND ANTIEPILEPTICS UNIV LAVAL (CA) 2019-09-11 EP disclosed
EP-2432776-B1 METHYL SULFANYL PYRIMIDINES USEFUL AS ANTIINFLAMMATORIES, ANALGESICS, AND ANTIEPILEPTICS UNIV LAVAL (CA) 2019-09-11 EP disclosed
CN-110023292-A Apoptosis inhibitor 北京生命科学研究所 2019-07-16 CN disclosed
WO-1995020572-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1995-08-03 WO disclosed
EP-0253766-B1 STABILIZED OLEFIN POLYMER INSULATING COMPOSITIONS CIBA-GEIGY AG (CH) 1992-03-11 EP disclosed
EP-0252878-B1 VOLTAGE STABILIZED POLYOLEFIN COMPOSITIONS AND SILICONE-GLYCOL DERIVATIVES SUITABLE THEREFOR CIBA-GEIGY AG (CH) 1990-11-22 EP disclosed
US-4724248-A POLYDIALKYLSILOXANEPOLYOXYALKYLENE BLOCK AND/OR GRAFT COPOLYMERS CIBA-GEIGY CORPORATION (US) 1988-02-09 US disclosed
EP-0253766-A2 Stabilized olefin polymer insulating compositions CIBA-GEIGY AG (CH) 1988-01-20 EP disclosed
EP-0252878-A1 Voltage stabilized polyolefin compositions and silicone-glycol derivatives suitable therefor CIBA-GEIGY AG (CH) 1988-01-13 EP disclosed
US-4689362-A POLYSILOXANE POLYOXYALKYLENE BLOCK OR GRAFT COPOLYMERS AS STABILIZERS CIBA-GEIGY CORPORATION (US) 1987-08-25 US disclosed
US-4268678-A 4-(Arylaliphatic)isoxazoles STERLING DRUG INC. (US) 1981-05-19 US disclosed
US-4171371-A Diketones STERLING DRUG INC. (US) 1979-10-16 US disclosed
US-4153719-A Aromatic diketones STERLING DRUG INC. (US) 1979-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11725000-B2 Apoptosis inhibitors BAX, SDHA, SDHB SLC6A4 3822/4885HTR2A 3517/4885KCNH2 3722/4885
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR SLC6A4 1160/4885HTR2A 134/4885KCNH2 1883/4885
US-11034680-B2 Apoptosis inhibitors BAX, SDHA, SDHB SLC6A4 3822/4885HTR2A 3517/4885KCNH2 3722/4885
US-20210309647-A1 Apoptosis Inhibitors BAX, SDHA, SDHB SLC6A4 3822/4885HTR2A 3517/4885KCNH2 3722/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.