SCHEMBL474017

SCHEMBL474017

Cn1c(=O)oc2ccc(CC(c3ccc(Oc4ncccn4)cc3Cl)C(O)C(F)(F)F)cc21

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 13/20 0.33
CYP11B2 P19099 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HSD17B10 Q99714 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
LMNA P02545 1/20 0.32
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473926 0.89 KMO (0.39) CYP11B2SMN1; SMN2LMNAMAPT
SCHEMBL474137 0.83 MIF (0.36) KCNJ1CYP11B2ALDH1A1MAPT
SCHEMBL474034 0.82 KMO (0.39) CYP11B2SMN1; SMN2LMNAMAPT
SCHEMBL473987 0.82 CYP11B2 (0.35) KCNJ1CYP11B2ALDH1A1NPC1MAPT
SCHEMBL474050 0.80 CYP11B2 (0.40) KCNJ1CYP11B2
SCHEMBL473936 0.79 CYP11B2 (0.45) KCNJ1CYP11B2
SCHEMBL473947 0.78 MIF (0.36) KCNJ1CYP11B2ALDH1A1LMNAMAPT
SCHEMBL474015 0.77 KDM4E (0.33) CYP11B2KDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL12164225 0.77 KDM4E (0.33) CYP11B2KDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL473924 0.75 CYP11B2 (0.41) CYP11B2KDM4EALDH1A1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed