SCHEMBL473926

SCHEMBL473926

COc1ccc(C(Cc2ccc3oc(=O)n(C)c3c2)C(O)C(F)(F)F)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.39
IDO1 P14902 1/20 0.37
MIF P14174 3/20 0.37
CD74 P04233 2/20 0.37
CBX7 O95931 4/20 0.35
CDYL2 Q8N8U2 4/20 0.35
CDYL Q9Y232 4/20 0.35
CDY1; CDY1B Q9Y6F8 4/20 0.35
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP11B2 P19099 1/20 0.34
LMNA P02545 2/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ASAH1 Q13510 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474034 0.93 KMO (0.39) KMOIDO1MIFCD74CBX7
SCHEMBL474017 0.89 KCNJ1 (0.33) CYP11B2LMNAMAPTSMN1; SMN2
SCHEMBL474137 0.88 MIF (0.36) IDO1MIFCD74KMT2ACYP11B2
SCHEMBL473987 0.87 CYP11B2 (0.35) IDO1KMT2ACYP11B2TP53MAPT
SCHEMBL473936 0.82 CYP11B2 (0.45) CYP11B2
SCHEMBL473947 0.82 MIF (0.36) IDO1MIFCD74KMT2ACYP11B2
SCHEMBL474050 0.81 CYP11B2 (0.40) CYP11B2
SCHEMBL473924 0.80 CYP11B2 (0.41) POLBKMT2ACYP11B2LMNAMAPT
SCHEMBL474062 0.78 CYP11B2 (0.35) KMOCYP11B2ASAH1
SCHEMBL12164174 0.74 KMO (0.38) KMOIDO1MIFCD74CBX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed