SCHEMBL473947

SCHEMBL473947

Cn1c(=O)oc2ccc(CC(c3cc(O)ccc3Cl)C(O)C(F)(F)F)cc21

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MIF P14174 4/20 0.36
CD74 P04233 2/20 0.36
CYP11B2 P19099 1/20 0.35
KCNJ1 P48048 3/20 0.34
IDO1 P14902 3/20 0.34
LRRK2 Q5S007 1/20 0.32
MAPT P10636 1/20 0.32
CTSC P53634 1/20 0.32
PKM P14618 1/20 0.31
GFER P55789 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474137 0.92 MIF (0.36) MIFCD74CYP11B2KCNJ1IDO1
SCHEMBL474034 0.88 KMO (0.39) MIFCD74CYP11B2IDO1MAPT
SCHEMBL473987 0.84 CYP11B2 (0.35) CYP11B2KCNJ1IDO1MAPTCTSC
SCHEMBL473926 0.82 KMO (0.39) MIFCD74CYP11B2IDO1MAPT
SCHEMBL474062 0.80 CYP11B2 (0.35) CYP11B2KCNJ1CTSC
SCHEMBL473936 0.79 CYP11B2 (0.45) CYP11B2KCNJ1CTSCGPR55
SCHEMBL474050 0.78 CYP11B2 (0.40) CYP11B2KCNJ1CTSCGPR55
SCHEMBL474017 0.78 KCNJ1 (0.33) CYP11B2KCNJ1MAPTALDH1A1LMNA
SCHEMBL473924 0.76 CYP11B2 (0.41) CYP11B2MAPTALDH1A1KMT2ALMNA
SCHEMBL12344679 0.73 KMO (0.38) MIFCYP11B2KCNJ1LRRK2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed