SCHEMBL474050

SCHEMBL474050

Cn1c(=O)oc2ccc(CC(c3ccc(-c4ccnnc4)cc3Cl)C(O)C(F)(F)F)cc21

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.40
KCNJ1 P48048 13/20 0.39
GPR55 Q9Y2T6 3/20 0.38
CTSC P53634 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473936 0.88 CYP11B2 (0.45) CYP11B2KCNJ1GPR55CTSC
SCHEMBL474137 0.83 MIF (0.36) CYP11B2KCNJ1CTSC
SCHEMBL473987 0.83 CYP11B2 (0.35) CYP11B2KCNJ1CTSC
SCHEMBL473926 0.81 KMO (0.39) CYP11B2
SCHEMBL474017 0.80 KCNJ1 (0.33) CYP11B2KCNJ1
SCHEMBL473947 0.78 MIF (0.36) CYP11B2KCNJ1GPR55CTSC
SCHEMBL473909 0.77 GPR55 (0.40) CYP11B2KCNJ1GPR55
SCHEMBL12164224 0.77 GPR55 (0.40) CYP11B2KCNJ1GPR55
SCHEMBL474034 0.76 KMO (0.39) CYP11B2
SCHEMBL473924 0.76 CYP11B2 (0.41) CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed