SCHEMBL4740409

SCHEMBL4740409

Cc1ccc(S(=O)(=O)N2CCCC(CC(=O)NN3CCCC(C)C3)C2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.47
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
KDM4E B2RXH2 2/20 0.45
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
MAPT P10636 3/20 0.44
TP53 P04637 3/20 0.44
THRB P10828 2/20 0.44
ALDH1A1 P00352 2/20 0.44
POLB P06746 2/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740197 0.91 LMNA (0.50) CYP19A1CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL4739834 0.87 CYP3A4 (0.61) CYP19A1CYP3A4CYP2C19KMT2AMEN1
SCHEMBL4738940 0.87 ALDH1A1 (0.53) CYP19A1CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL4782859 0.84 SMN1; SMN2 (0.50) CYP19A1CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL4739879 0.81 RAB9A (0.58) KDM4EKMT2AMEN1MAPTTP53
SCHEMBL4738947 0.79 CYP3A4 (0.64) CYP19A1CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL4738938 0.78 TSHR (0.56) CYP19A1KMT2AMEN1MAPTTP53
SCHEMBL4740145 0.78 MAPT (0.49) CYP19A1CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL4740901 0.78 CYP19A1 (0.58) CYP19A1CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL4740148 0.78 TSHR (0.50) KMT2AMEN1TP53POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO disclosed