SCHEMBL474057

SCHEMBL474057

CC(c1c(C(=O)O)cccc1-c1ccccc1)C(O)(c1ccc2oc(=O)n(C)c2c1)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
ASAH1 Q13510 2/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
CMA1 P23946 2/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
CTSG P08311 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2C9 P11712 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SCD5 Q86SK9 1/20 0.32
CYP11B2 P19099 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473961 0.94 ALDH1A1 (0.41) ASAH1ALDH1A1HPGDCMA1MAPT
SCHEMBL474521 0.85 TP53 (0.39) NR1H3ALDH1A1CMA1SMN1; SMN2
SCHEMBL474051 0.82 ALDH1A1 (0.39) KMOASAH1ALDH1A1HPGDMAPT
SCHEMBL473903 0.77 ALDH1A1 (0.37) NR1H2NR1H3ALDH1A1CMA1MAPT
SCHEMBL12164103 0.76 GPR55 (0.36) KMOMAPTTHRBSMN1; SMN2CYP11B2
SCHEMBL473904 0.76 ALDH1A1 (0.46) ASAH1ALDH1A1HPGDMAPTTHRB
SCHEMBL2817228 0.74 GPR55 (0.36) KMOASAH1MAPTSMN1; SMN2CYP11B2
SCHEMBL15520687 0.74 GPR55 (0.36) KMOASAH1MAPTSMN1; SMN2CYP11B2
SCHEMBL473893 0.74 KMO (0.36) KMOASAH1CMA1CTSGCYP2C8
SCHEMBL12164099 0.74 GPR55 (0.36) KMOMAPTCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed