SCHEMBL4744588

SCHEMBL4744588

CCC(CC)NC(=O)Nc1ccc(Oc2ccc(NC(=O)O)c(F)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.57
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
TAS1R3 Q7RTX0 1/20 0.48
TAS1R1 Q7RTX1 1/20 0.48
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
SLC1A3 P43003 1/20 0.45
SLC1A2 P43004 1/20 0.45
SLC1A1 P43005 1/20 0.45
HPGD P15428 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
MAPK1 P28482 1/20 0.44
HRH3 Q9Y5N1 3/20 0.43
MAPT P10636 1/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MTNR1B P49286 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688990 0.87 PKM (0.50) PKMTAS1R3TAS1R1NPC1RAB9A
SCHEMBL4683259 0.86 PKM (0.49) PKMTAS1R3TAS1R1NPC1RAB9A
SCHEMBL4236455 0.84 PKM (0.63) PKMTAS1R3TAS1R1NPC1RAB9A
SCHEMBL4785963 0.84 PKM (0.63) PKMTAS1R3TAS1R1NPC1RAB9A
SCHEMBL4233255 0.84 PKM (0.59) PKMCYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL4744778 0.82 PKM (0.52) PKMCYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL4240208 0.81 PKM (0.63) PKMTAS1R3TAS1R1NPC1RAB9A
SCHEMBL4689054 0.81 TAS1R3 (0.72) PKMCYP2C9CYP2C19TAS1R3TAS1R1
SCHEMBL4240960 0.80 PKM (0.58) PKMTAS1R3TAS1R1NPC1RAB9A
SCHEMBL4240206 0.80 PKM (0.60) PKMTAS1R3TAS1R1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP disclosed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO disclosed