SCHEMBL4745700

SCHEMBL4745700

CC(C)COC(=O)N1CCc2cc(-c3cnc4[nH]cc(C#N)c4c3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
PAK1 Q13153 3/20 0.42
CYP11B1 P15538 7/20 0.42
CYP11B2 P19099 6/20 0.42
PKN1 Q16512 1/20 0.42
AAK1 Q2M2I8 2/20 0.39
MAP3K12 Q12852 2/20 0.38
GPR119 Q8TDV5 1/20 0.38
RET P07949 1/20 0.38
NPC1 O15118 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
USP2 O75604 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14069149 0.85 BRD4 (0.46) PRMT5WDR77PAK1CYP11B1CYP11B2
SCHEMBL2373579 0.70 RORC (0.40) CYP11B1CYP11B2GPR119NPC1ALDH1A1
SCHEMBL2373819 0.69 ABHD6 (0.59) GPR119NPC1RAB9ASMN1; SMN2GFER
SCHEMBL4747825 0.68 PRMT5 (0.49) PRMT5WDR77CYP11B1CYP11B2AAK1
SCHEMBL2373645 0.67 RIPK1 (0.68)
SCHEMBL4746507 0.66 DYRK1A (0.56) PRMT5WDR77AAK1
SCHEMBL4200987 0.66 MAPK8 (0.60) PRMT5WDR77AAK1MAP3K12
SCHEMBL4743697 0.66 PRMT5 (0.53) PRMT5WDR77AAK1
SCHEMBL2778816 0.66 NPC1 (0.64) PRMT5WDR77NPC1ALDH1A1MAPT
SCHEMBL4747758 0.66 PRMT5 (0.55) PRMT5WDR77AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO claimed
WO-2008110508-A1 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH INAPPROPRIATE IKK1 ACTIVITY GLAXO GROUP LIMITED (GB) 2008-09-18 WO disclosed