SCHEMBL2373579

SCHEMBL2373579

CC(C)COC(=O)N1CCc2cc(-c3cccc(F)c3C#N)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.40
CYP11B1 P15538 7/20 0.39
CYP11B2 P19099 6/20 0.39
USP30 Q70CQ3 1/20 0.39
SCN9A Q15858 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GPR119 Q8TDV5 2/20 0.38
EIF2AK3 Q9NZJ5 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL869258 0.83 BRD4 (0.47) RORCCYP11B1CYP11B2USP30NPC1
SCHEMBL2374644 0.75 KDR (0.43) CYP11B1CYP11B2EIF2AK3RIPK1
SCHEMBL2373984 0.73 NOTUM (0.60) SCN9ASCN10ANPC1RAB9AL3MBTL1
SCHEMBL2373819 0.73 ABHD6 (0.59) HTR2ANPC1RAB9AL3MBTL1GPR119
SCHEMBL2778816 0.72 NPC1 (0.64) NPC1RAB9AL3MBTL1ALDH1A1MAPT
SCHEMBL4745700 0.70 PRMT5 (0.43) CYP11B1CYP11B2NPC1RAB9AGPR119
SCHEMBL5269117 0.69 GPR119 (0.41) NPC1RAB9AL3MBTL1GPR119ALDH1A1
SCHEMBL2375097 0.69 EIF2AK3 (0.65) NPC1RAB9AEIF2AK3ALDH1A1MAPT
SCHEMBL2373042 0.67 EIF2AK3 (0.43) NPC1RAB9AGPR119EIF2AK3ALDH1A1
SCHEMBL2373645 0.67 RIPK1 (0.68) EIF2AK3RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2549868-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2013-01-30 EP disclosed
WO-2011119663-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed