SCHEMBL4746475

SCHEMBL4746475

CCOC(=O)c1cc(C(=O)O)cc(-c2cccnc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
MAPT P10636 3/20 0.57
CYP2C9 P11712 2/20 0.57
CYP2C19 P33261 2/20 0.57
KMO O15229 1/20 0.57
MMP2 P08253 1/20 0.56
MMP13 P45452 1/20 0.56
MMP14 P50281 1/20 0.56
MKNK1 Q9BUB5 2/20 0.52
MKNK2 Q9HBH9 2/20 0.52
KDM4E B2RXH2 3/20 0.49
NPSR1 Q6W5P4 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28143431 0.85 KMO (0.61) ALDH1A1MAPTKMOMKNK1MKNK2
SCHEMBL1895643 0.85 CYP2C9 (0.57) ALDH1A1MAPTCYP2C9CYP2C19KMO
SCHEMBL15557036 0.84 CYP2C9 (0.55) CYP2C9CYP2C19CYP1A2NPC1RAB9A
SCHEMBL17089048 0.84 KMO (0.77) ALDH1A1MAPTKMOMKNK1MKNK2
SCHEMBL29503876 0.84 KMO (0.77) ALDH1A1MAPTKMOMKNK1MKNK2
SCHEMBL10028690 0.84 ALDH1A1 (0.56) ALDH1A1MAPTCYP2C9CYP2C19KMO
SCHEMBL5735824 0.82 MKNK1 (0.59) ALDH1A1MAPTCYP2C9CYP2C19MMP2
SCHEMBL10028699 0.81 KMO (0.77) ALDH1A1MAPTKMOMKNK1MKNK2
SCHEMBL14395132 0.80 KMO (0.67) ALDH1A1KMOMKNK1MKNK2KDM4E
SCHEMBL3510029 0.80 RAB9A (0.57) ALDH1A1MAPTCYP2C9CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008119773-A1 AMIDE DERIVATIVES AS INHIBITORS OF ASPARTYL PROTEASES MEDIVIR AB (SE) 2008-10-09 WO disclosed