SCHEMBL4746538

SCHEMBL4746538

C[C@H](c1ccc(F)cc1F)N1C(=O)c2cc(Br)cc(N)c2C1=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
HSD11B1 P28845 1/20 0.34
ALDH1A1 P00352 1/20 0.32
APLNR P35414 2/20 0.31
SIGMAR1 Q99720 1/20 0.31
OPRM1 P35372 1/20 0.30
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746540 1.00 IDO1 (0.34) IDO1TDO2HSD11B1ALDH1A1APLNR
SCHEMBL4746488 0.78 HSD11B1 (0.39) HSD11B1SIGMAR1OPRM1
SCHEMBL4746505 0.78 HSD11B1 (0.39) HSD11B1SIGMAR1OPRM1
SCHEMBL4748815 0.78 HSD11B1 (0.39) HSD11B1SIGMAR1OPRM1
SCHEMBL4746487 0.78 HSD11B1 (0.39) HSD11B1SIGMAR1OPRM1
SCHEMBL4749155 0.77 AAK1 (0.36)
SCHEMBL4749154 0.77 AAK1 (0.36)
SCHEMBL4831699 0.72 OPRM1 (0.46) ALDH1A1APLNROPRM1
SCHEMBL4788355 0.70 HSD11B1 (0.44) IDO1TDO2HSD11B1SIGMAR1CES2
SCHEMBL31145949 0.68 HSD11B1 (0.43) IDO1TDO2HSD11B1SIGMAR1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124518-A1 OXO-DIHYDROISOINDOLE SULFONAMIDE COMPOUNDS AS MODULATORS OF THE CCK2 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2008-10-16 WO disclosed