SCHEMBL4747779

SCHEMBL4747779

NC(=O)c1ccc([N+](=O)[O-])c(-c2ccc(O)cc2)c1-c1ccc(O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HIF1A Q16665 1/20 0.40
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 5/20 0.39
MEN1 O00255 3/20 0.39
GAA P10253 2/20 0.39
ERN1 O75460 1/20 0.38
BACE1 P56817 2/20 0.37
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37
PARP1 P09874 1/20 0.36
CASP1 P29466 1/20 0.36
POLB P06746 2/20 0.36
TDP1 Q9NUW8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7064896 0.83 ESR1 (0.43) TSHRHPGDALDH1A1LMNAMAPT
SCHEMBL11367351 0.75 BACE1 (0.49) CYP3A4KMT2AALDH1A1LMNAMAPT
SCHEMBL1883040 0.75 MAPT (0.49) CYP3A4TSHRSMN1; SMN2KMT2AALDH1A1
SCHEMBL30029048 0.75 ALDH1A1 (0.40) CYP3A4TSHRTP53HPGDSMN1; SMN2
SCHEMBL27462702 0.75 MAPT (0.43) CYP3A4TSHRKMT2AALDH1A1LMNA
SCHEMBL27376059 0.74 GPR35 (0.57) CYP3A4TSHRTP53HPGDSMN1; SMN2
SCHEMBL27607677 0.74 MEN1 (0.45) CYP3A4TSHRTP53HPGDSMN1; SMN2
SCHEMBL4750554 0.73 DGAT1 (0.41) TSHRHPGDALDH1A1MAPTERN1
SCHEMBL299878 0.73 FBP1 (0.49) CYP3A4TSHRTP53ALDH1A1PARP1
SCHEMBL27271193 0.73 ALDH1A1 (0.47) CYP3A4TSHRSMN1; SMN2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130571-A1 NUCLEAR RECEPTOR BINDING AGENTS GTX, INC. (US) 2008-10-30 WO disclosed