SCHEMBL474936

SCHEMBL474936

CC(c1ccccc1-c1ccc(OCC(=O)O)cc1)C(O)(c1ccc2c(c1)n(C)c(=O)n2C)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.42
ADORA2B P29275 10/20 0.42
PTGDR2 Q9Y5Y4 3/20 0.38
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
BRD4 O60885 1/20 0.36
BRPF1 P55201 1/20 0.36
ADORA1 P30542 2/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
SRD5A2 P31213 1/20 0.35
PPARG P37231 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474933 0.91 PPARG (0.39) ADORA2AADORA2BPTGDR2PPARDSMN1; SMN2
SCHEMBL474397 0.85 ADORA2A (0.42) ADORA2AADORA2BPPARDPPARASMN1; SMN2
SCHEMBL12164042 0.82 SMN1; SMN2 (0.40) ADORA2AADORA2BPPARDSMN1; SMN2BRD4
SCHEMBL474253 0.82 SMN1; SMN2 (0.40) ADORA2AADORA2BPPARDSMN1; SMN2BRD4
SCHEMBL474976 0.82 PTGDR2 (0.39) PTGDR2PPARDPPARASMN1; SMN2BRPF1
SCHEMBL474296 0.80 TRIM24 (0.47) ADORA2AADORA2BPPARDPPARASMN1; SMN2
SCHEMBL12164048 0.80 TRIM24 (0.47) ADORA2AADORA2BPPARDPPARASMN1; SMN2
SCHEMBL474633 0.78 ALDH1A1 (0.41) SMN1; SMN2BRD4BRPF1
SCHEMBL474975 0.76 ALDH1A1 (0.35) PTGDR2SMN1; SMN2
SCHEMBL474521 0.75 TP53 (0.39) SMN1; SMN2BRPF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed