SCHEMBL474975

SCHEMBL474975

CC(c1c(CC(=O)O)cccc1-c1ccccc1)C(O)(c1ccc2c(c1)n(C)c(=O)n2C)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GLA P06280 1/20 0.35
PTGS2 P35354 2/20 0.35
MAPK14 Q16539 2/20 0.35
CMA1 P23946 5/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
GAA P10253 1/20 0.33
PTGS1 P23219 1/20 0.33
TRPA1 O75762 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
GRM2 Q14416 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474521 0.86 TP53 (0.39) ALDH1A1SMN1; SMN2GLAMAPK14CMA1
SCHEMBL474976 0.82 PTGDR2 (0.39) ALDH1A1SMN1; SMN2GLAPTGS2MAPK14
SCHEMBL474483 0.81 SMN1; SMN2 (0.35) ALDH1A1SMN1; SMN2GLAPTGS2MAPK14
SCHEMBL474633 0.77 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2GLAMAPK14CMA1
SCHEMBL474936 0.76 ADORA2A (0.42) SMN1; SMN2PTGDR2
SCHEMBL474933 0.76 PPARG (0.39) ALDH1A1SMN1; SMN2PTGDR2PDCD1CD274
SCHEMBL12164010 0.76 PTGS2 (0.37) ALDH1A1PTGS2CMA1PTGDR2GRM2
SCHEMBL474492 0.76 PTGS2 (0.37) ALDH1A1PTGS2CMA1PTGDR2GRM2
SCHEMBL473961 0.73 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2CMA1
SCHEMBL474606 0.72 RXRA (0.40) ALDH1A1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed