SCHEMBL4749974

SCHEMBL4749974

NC1COc2cccc(OS(=O)(=O)c3cccnc3)c2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.35
METAP1 P53582 1/20 0.35
NAPRT Q6XQN6 1/20 0.34
CYP19A1 P11511 1/20 0.33
HPGD P15428 3/20 0.33
SCN9A Q15858 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SCN5A Q14524 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 2/20 0.33
F2 P00734 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CA9 Q16790 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
DRD2 P14416 1/20 0.32
ADRA1D P25100 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749973 1.00 METAP2 (0.35) METAP2METAP1NAPRTCYP19A1HPGD
SCHEMBL4788147 0.78 SCN9A (0.44) SCN9ASCN5A
SCHEMBL4788156 0.78 SCN9A (0.44) SCN9ASCN5A
SCHEMBL4788597 0.73 CNR2 (0.36) ALDH1A1DRD2
SCHEMBL4788607 0.73 CNR2 (0.36) ALDH1A1DRD2
SCHEMBL4789099 0.73 HTR1A (0.31) DRD2HTR1A
SCHEMBL4789100 0.73 HTR1A (0.31) DRD2HTR1A
SCHEMBL841717 0.71 SCN9A (0.50) CYP19A1HPGDSCN9AALDH1A1SCN5A
Ammonia Solution, Strong SCHEMBL3672627 0.70 SCN9A (0.49) CYP19A1HPGDSCN9AALDH1A1SCN5A
SCHEMBL4839911 0.70 DRD2 (0.54) DRD2ADRA1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130319-A2 NOVEL N-TETRAHYDRONAPHTALENE OR N-CHROMANE CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed