SCHEMBL4749987

SCHEMBL4749987

COc1ccc(-n2ccc3cc(C(C)C)nc(N4CCCCC4)c3c2=O)cc1OC

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.42
HIF1A Q16665 3/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
GAA P10253 1/20 0.36
THRB P10828 1/20 0.36
HTR2C P28335 2/20 0.36
MCHR1 Q99705 2/20 0.36
LPAR5 Q9H1C0 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAP2K7 O14733 1/20 0.35
HTR2B P41595 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4907061 0.84 EGFR (0.42) EGFRHIF1AMEN1KMT2AALDH1A1
SCHEMBL4747371 0.83 NPC1 (0.34) EGFRMEN1KMT2AALDH1A1MAPT
SCHEMBL5813982 0.77 SYK (0.39) ALDH1A1MAPTKDM4EHPGDGAA
SCHEMBL5814919 0.76 KDM5A (0.33) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL4788702 0.74 GRM2 (0.36) MEN1KMT2AMAPTKDM4EPOLB
SCHEMBL5816427 0.74 GRM2 (0.35) ALDH1A1MAPTKDM4EHPGD
SCHEMBL5821178 0.70 HIF1A (0.39) HIF1AMEN1KMT2AALDH1A1MAPT
SCHEMBL4750208 0.68 JAK2 (0.43) ALDH1A1MAPTKDM4EHPGD
SCHEMBL5820228 0.67 KCNH2 (0.39) EGFRMEN1KMT2AALDH1A1MAPT
SCHEMBL28860292 0.67 ALDH1A1 (0.63) HIF1AMEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO disclosed