SCHEMBL4750217

SCHEMBL4750217

CCn1ccc2cc(C)nc(C3CCCCC3)c2c1=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.37
GRM2 Q14416 3/20 0.35
MAT2A P31153 2/20 0.34
ADORA1 P30542 3/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
SRC P12931 1/20 0.33
CHRM4 P08173 1/20 0.33
FAAH O00519 1/20 0.33
SPR P35270 1/20 0.32
CTSK P43235 3/20 0.32
CTSS P25774 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4747715 0.99 PDE2A (0.37) PDE2AGRM2MAT2AADORA1ALDH1A1
SCHEMBL4747767 0.94 GRM2 (0.37) PDE2AGRM2SRC
SCHEMBL4750004 0.77 GRM2 (0.39) GRM2ALDH1A1
SCHEMBL4750623 0.76 GRM2 (0.40) GRM2ALDH1A1
SCHEMBL4747299 0.74 GRM2 (0.38) GRM2ALDH1A1
SCHEMBL4747263 0.72 GRM2 (0.36) GRM2ALDH1A1
SCHEMBL4750023 0.67 HSF1 (0.41) GRM2MAT2AADORA1ALDH1A1POLB
SCHEMBL10232910 0.66 KDM4E (0.41) GRM2ALDH1A1
SCHEMBL4788109 0.66 MAPK9 (0.44) ADORA1ALDH1A1POLB
SCHEMBL4747717 0.65 GRM2 (0.36) GRM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed