SCHEMBL4750221

SCHEMBL4750221

Cc1cc2c(c(-c3ccc(F)cc3)n1)C(=O)NCC2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RIPK3 Q9Y572 13/20 0.45
PARP10 Q53GL7 3/20 0.44
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
GABRA5 P31644 2/20 0.44
PARP1 P09874 1/20 0.44
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
PARP11 Q9NR21 2/20 0.43
GRM5 P41594 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072395 0.76 NPC1 (0.39)
SCHEMBL4751106 0.75 GABRG2 (0.41) GABRG2GABRB3GABRA5
SCHEMBL4747756 0.73 HRH3 (0.39)
SCHEMBL4785722 0.72 ALDH1A1 (0.41)
SCHEMBL4251098 0.71 ADORA2A (0.35)
SCHEMBL4747297 0.70 HRH3 (0.42) RIPK3GABRG2GABRB3GABRA5
SCHEMBL4788529 0.69 HTR2A (0.38)
SCHEMBL4786612 0.69 ALDH1A1 (0.39)
SCHEMBL4750242 0.69 HRH3 (0.58)
SCHEMBL4750215 0.69 PDGFRB (0.42) GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed