SCHEMBL4751256

SCHEMBL4751256

O=C1CN(C(=O)c2ccc(Cl)cc2)CCN1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.55
HRH3 Q9Y5N1 1/20 0.54
POLB P06746 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 1/20 0.52
RAB9A P51151 1/20 0.52
PHGDH O43175 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MDM2 Q00987 6/20 0.50
MAPK14 Q16539 1/20 0.48
MAPT P10636 1/20 0.48
MGLL Q99685 1/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21170645 0.84 HRH3 (0.54) HSP90AA1HRH3POLBTDP1SMN1; SMN2
SCHEMBL14117676 0.84 HRH3 (0.54) HSP90AA1HRH3POLBTDP1RAB9A
SCHEMBL12093445 0.84 PKM (0.67) HSP90AA1HRH3POLBTDP1GAA
SCHEMBL10883109 0.84 SIGMAR1 (0.62) HSP90AA1HRH3POLBTDP1RAB9A
SCHEMBL12090013 0.84 ALDH1A1 (0.57) HSP90AA1HRH3POLBTDP1SMN1; SMN2
SCHEMBL106697 0.84 HPGD (0.59) HSP90AA1HRH3POLBTDP1SMN1; SMN2
SCHEMBL9971990 0.83 HSP90AA1 (0.54) HSP90AA1HRH3POLBTDP1SMN1; SMN2
SCHEMBL9971981 0.82 PKM (0.54) HSP90AA1POLBTDP1SMN1; SMN2GAA
SCHEMBL105677 0.80 HSP90AA1 (0.57) HSP90AA1POLBTDP1SMN1; SMN2GAA
SCHEMBL10008491 0.80 HPGD (0.56) HRH3POLBTDP1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008136754-A1 NOVEL BENZYL - 2 -OXO-PIPERAZINYL/ 7-OXO/5-OXA- [1,4] DIAZEPANYL/ 2 -OXO- TETRAHYDROPYRIMIDINYL DERIVATIVES ASTRAZENECA AB (SE) 2008-11-13 WO disclosed