SCHEMBL4751580

SCHEMBL4751580

Cc1c(F)cccc1C1C(C(=O)c2cccc(O)c2F)CN(CCCCN(C)C)CC1C(=O)[C@@H]1CN(CCCCN(C)C)C[C@H](C(=O)c2cccc(O)c2F)[C@@H]1c1cccc(F)c1C

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.35
ACHE P22303 1/20 0.35
HRH2 P25021 1/20 0.32
HRH1 P35367 1/20 0.32
HSP90B1 P14625 1/20 0.32
TRAP1 Q12931 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31
MGLL Q99685 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749430 1.00 KIF11 (0.35) KIF11ACHEHRH2HRH1HSP90B1
SCHEMBL4752017 0.89 KIF11 (0.40) KIF11ACHEKDM4E
SCHEMBL4749443 0.88 PIN1 (0.36) KIF11ACHEHSP90B1TRAP1KDM4E
SCHEMBL4749425 0.88 PIN1 (0.36) KIF11ACHEHSP90B1TRAP1KDM4E
SCHEMBL4749258 0.87 KIF11 (0.35) KIF11ACHEHSP90B1TRAP1MGLL
SCHEMBL4749270 0.87 KIF11 (0.35) KIF11ACHEHSP90B1TRAP1MGLL
SCHEMBL4751821 0.85 MEN1 (0.36) KIF11ACHEHSP90B1TRAP1KDM4E
SCHEMBL4019728 0.85 TAS1R3 (0.36) HRH2HRH1TAS1R3TAS1R1TAS1R2
SCHEMBL4027811 0.85 KDM1A (0.34) TAS1R3TAS1R1TAS1R2
SCHEMBL4749505 0.84 KIF11 (0.35) KIF11ACHEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO claimed
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO disclosed