SCHEMBL4752010

SCHEMBL4752010

Cc1c(F)cccc1C1[C@@H](C(=O)c2cccc(O)c2)CN(C2CN3CCC2CC3)C[C@@H]1C(=O)c1cccc(O)c1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
MGLL Q99685 6/20 0.36
CHRNA7 P36544 4/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
HTR3A P46098 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752021 1.00 ALDH1A1 (0.38) ALDH1A1MGLLCHRNA7CHRNB2CHRNB4
SCHEMBL4749213 0.88 ALDH1A1 (0.32) ALDH1A1MGLL
SCHEMBL4749216 0.88 ALDH1A1 (0.32) ALDH1A1MGLL
SCHEMBL4019273 0.83 MGLL (0.35) MGLL
SCHEMBL4018836 0.83 GRIN1 (0.38) MGLL
SCHEMBL4029076 0.83 MGLL (0.35) MGLL
SCHEMBL4751751 0.82 MGLL (0.39) ALDH1A1MGLL
SCHEMBL4749392 0.82 MGLL (0.36) MGLL
SCHEMBL4751750 0.82 MGLL (0.39) ALDH1A1MGLL
SCHEMBL4021646 0.82 MC4R (0.36) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO disclosed