SCHEMBL4754478

SCHEMBL4754478

C(=CC1CCNCC1)c1cncc(OCC2CC2)c1.C(=CC1CNC1)c1cncnc1.CN1CCC(C=Cc2ccc(Cl)nc2)CC1.CN1CCC(C=Cc2cncc(OCC3CC3)c2)CC1.Clc1ccc(C=CC2CCNCC2)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA3 P32297 5/20 0.37
CHRNB1 P11230 4/20 0.37
CHRNB2 P17787 4/20 0.37
CHRNB4 P30926 4/20 0.37
CHRNB3 Q05901 4/20 0.37
AKT1 P31749 5/20 0.35
CHUK O15111 1/20 0.32
DYRK3 O43781 1/20 0.32
ROCK2 O75116 1/20 0.32
MAP4K4 O95819 1/20 0.32
PIM1 P11309 1/20 0.32
PRKACA P17612 1/20 0.32
RPS6KB1 P23443 1/20 0.32
CLK2 P49760 1/20 0.32
PRKX P51817 1/20 0.32
PRKG2 Q13237 1/20 0.32
ROCK1 Q13464 1/20 0.32
DYRK1A Q13627 1/20 0.32
PRKG1 Q13976 1/20 0.32
PKN2 Q16513 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6102061 0.94 CHRNB1 (0.36) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL6102057 0.94 CHRNB1 (0.36) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL1645371 0.86 CHRNB2 (0.39) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL6225866 0.86 CHRNB1 (0.44) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL2214137 0.83 AKT1 (0.42) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL2214139 0.83 AKT1 (0.42) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL2214142 0.83 AKT1 (0.42) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL1349334 0.80 CHRNB2 (0.49) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL1349331 0.80 CHRNB2 (0.49) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3
SCHEMBL1349085 0.78 AKT1 (0.50) CHRNA3CHRNB1CHRNB2CHRNB4CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157365-A2 VINYLAZACYCLOALKANES FOR TREATING NEUROPATHIC PAIN TARGACEPT, INC. (US) 2008-12-24 WO disclosed