SCHEMBL4754879

SCHEMBL4754879

COCn1c(C)nc2c(Cl)ccnc21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.40
KDM4E B2RXH2 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ALDH1A1 P00352 2/20 0.33
PDE4B Q07343 1/20 0.33
DCTPP1 Q9H773 1/20 0.33
PDE10A Q9Y233 2/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22438726 0.79 DCTPP1 (0.54) HTR6KDM4ESMN1; SMN2ALDH1A1DCTPP1
SCHEMBL25297700 0.74 NR3C1 (0.37) HTR6KDM4EALDH1A1HTT
SCHEMBL4753554 0.74 PDE10A (0.32) HSD17B10PDE10A
SCHEMBL4751475 0.71 CDK4 (0.32) DCTPP1
SCHEMBL6821486 0.70 CYP1A2 (0.46) HSD17B10ALDH1A1PDE4BPDE10A
SCHEMBL20163948 0.69 HTR6 (0.33) HTR6KDM4EPDE4B
SCHEMBL31240613 0.69 CDC7 (0.33) KDM4ESMN1; SMN2ALDH1A1
SCHEMBL2039524 0.69 CDC7 (0.33) KDM4ESMN1; SMN2ALDH1A1
SCHEMBL18359503 0.67 PIK3CD (0.46)
SCHEMBL24615302 0.66 MAPT (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008144253-A1 PROTEIN KINASE INHIBITORS AND METHODS FOR USING THEREOF IRM LLC (BM) 2008-11-27 WO disclosed
WO-2008144253-A1 PROTEIN KINASE INHIBITORS AND METHODS FOR USING THEREOF IRM LLC (BM) 2008-11-27 WO disclosed