SCHEMBL4755117

SCHEMBL4755117

CCOC(=O)CC(C[N+](=O)[O-])c1cc(Cl)cc(C(=O)OCC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
LMNA P02545 2/20 0.38
KMT2A Q03164 2/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA14 Q9ULX7 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
TRPV1 Q8NER1 1/20 0.35
F10 P00742 4/20 0.35
F2 P00734 3/20 0.35
PRSS1 P07477 1/20 0.35
ALDH1A1 P00352 3/20 0.34
RAB9A P51151 2/20 0.34
PKM P14618 1/20 0.34
CRHBP P24387 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31115525 0.82 F2 (0.47) NPC1LMNAKMT2ACA12CA1
SCHEMBL563397 0.81 F10 (0.43) NPC1LMNAKMT2AMEN1MAPT
SCHEMBL657923 0.80 MAPT (0.46) LMNAKMT2ACA12CA1CA2
SCHEMBL20475329 0.78 MAPT (0.41) NPC1LMNAMAPTKDM4EF10
SCHEMBL7682360 0.77 L3MBTL1 (0.42) LMNAKMT2AMEN1MAPTALDH1A1
SCHEMBL15548874 0.77 MAPT (0.40) LMNAKMT2AMEN1MAPTKDM4E
SCHEMBL9294262 0.75 F2 (0.50) NPC1LMNAKMT2AMEN1MAPT
SCHEMBL20475355 0.75 MAPT (0.39) LMNAKMT2AMEN1MAPTKDM4E
SCHEMBL20475388 0.75 KDM4E (0.44) LMNAKMT2AMEN1MAPTKDM4E
SCHEMBL6556296 0.74 ALDH1A1 (0.44) LMNAKMT2AMEN1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed