SCHEMBL4755507

SCHEMBL4755507

O=C(NCCNCc1ccc(Oc2ccccc2)cc1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.64
MAPK14 Q16539 5/20 0.63
CA12 O43570 1/20 0.60
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
MMP2 P08253 1/20 0.60
CA9 Q16790 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.59
LMNA P02545 2/20 0.59
CYP3A4 P08684 1/20 0.59
HTT P42858 1/20 0.59
MMP13 P45452 1/20 0.59
OPRM1 P35372 1/20 0.56
OPRD1 P41143 1/20 0.56
OPRK1 P41145 1/20 0.56
EPHX2 P34913 2/20 0.54
PPARG P37231 1/20 0.54
PPARA Q07869 1/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3038826 0.93 HPGD (0.63) HPGDMAPK14CA12CA1CA2
SCHEMBL3039071 0.91 EPHX2 (0.64) HPGDMAPK14CA12CA1CA2
SCHEMBL3035490 0.88 HPGD (0.56) HPGDMAPK14CA12CA1CA2
SCHEMBL5709300 0.86 HPGD (0.84) HPGDMAPK14SMN1; SMN2LMNACYP3A4
SCHEMBL8851840 0.86 ALDH1A1 (0.64) HPGDSMN1; SMN2LMNAEPHX2NPC1
SCHEMBL3035704 0.83 XDH (0.61) HPGDMAPK14CA12CA1CA2
SCHEMBL3043398 0.81 ADRB1 (0.56) HPGDMAPK14CA12CA1CA2
SCHEMBL27601039 0.81 NAAA (0.63) HPGDMAPK14CA12CA1CA2
SCHEMBL3043353 0.81 FAAH (0.51) HPGDMAPK14SMN1; SMN2LMNACYP3A4
SCHEMBL8738317 0.80 HPGD (0.97) HPGDMAPK14SMN1; SMN2LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976828-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Schering Aktiengesellschaft (DE) 2008-10-08 EP claimed
WO-2007079078-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-07-12 WO claimed
EP-1976828-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Schering Aktiengesellschaft (DE) 2008-10-08 EP disclosed
WO-2007079078-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-07-12 WO disclosed