SCHEMBL4755635

SCHEMBL4755635

O=c1cc(CO)nc([C@H]2CC[C@@H](C(F)(F)F)CC2)n1-c1ccc(Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.38
NOTUM Q6P988 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
DRD1 P21728 2/20 0.34
DRD5 P21918 2/20 0.34
MCHR1 Q99705 3/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AOC2 O75106 1/20 0.34
KCNH2 Q12809 3/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
POLB P06746 1/20 0.33
TP53 P04637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
GRM5 P41594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755639 1.00 AVPR1A (0.38) AVPR1ANOTUMKDM4EMAPTDRD1
SCHEMBL13985415 0.93 AVPR1A (0.36) AVPR1ANOTUMKDM4EMAPTDRD1
SCHEMBL4755622 0.90 AVPR1A (0.37) AVPR1ADRD1DRD5MCHR1LMNA
SCHEMBL4755627 0.90 AVPR1A (0.37) AVPR1ADRD1DRD5MCHR1LMNA
SCHEMBL13985226 0.89 TBK1 (0.33) AVPR1AKCNH2DRD2DRD3
SCHEMBL13985528 0.87 MCHR1 (0.38) AVPR1AMAPTDRD1DRD5MCHR1
SCHEMBL13985227 0.86 NOTUM (0.39) NOTUMKCNH2DRD2DRD3
SCHEMBL4753779 0.86 MCHR1 (0.35) AVPR1ADRD1DRD5MCHR1LMNA
SCHEMBL4753777 0.86 MCHR1 (0.35) AVPR1ADRD1DRD5MCHR1LMNA
SCHEMBL13985427 0.85 AVPR1A (0.34) AVPR1ADRD1DRD5MCHR1AOC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed