SCHEMBL4755677

SCHEMBL4755677

CN1CCN(c2cc(Cl)cc(-c3nnc(CC(=O)O)o3)c2)CC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 8/20 0.54
GAA P10253 1/20 0.46
CYP1B1 Q16678 2/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
DGAT1 O75907 3/20 0.39
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756936 0.88 CALCRL (0.53) CALCRLGAAMAPTSMN1; SMN2DGAT1
SCHEMBL4758257 0.82 RXRA (0.43) CALCRLMAPTSMN1; SMN2MEN1USP2
SCHEMBL13985180 0.76 SMN1; SMN2 (0.53) CALCRLGAAMAPTSMN1; SMN2POLB
SCHEMBL4758251 0.76 CALCRL (0.46) CALCRLMAPTSMN1; SMN2MEN1USP2
SCHEMBL4757912 0.75 RXRA (0.38) CALCRLMAPTSMN1; SMN2
SCHEMBL4757784 0.75 CALCRL (0.53) CALCRLMAPTSMN1; SMN2
SCHEMBL4755690 0.74 CALCRL (0.40) CALCRLMAPTSMN1; SMN2
SCHEMBL4756909 0.74 RXRA (0.37) CALCRLSMN1; SMN2
SCHEMBL4757909 0.74 CALCRL (0.73) CALCRL
SCHEMBL4755125 0.73 TP53 (0.45) CALCRLMAPTSMN1; SMN2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed