SCHEMBL4755763

SCHEMBL4755763

CNc1nc(C2CCC(C(F)(F)F)CC2)n(-c2ccc(Cl)nc2)c(=O)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.36
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
YTHDC1 Q96MU7 1/20 0.32
LRRK2 Q5S007 1/20 0.32
APLNR P35414 1/20 0.31
CHRM4 P08173 1/20 0.31
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31
DRD1 P21728 2/20 0.31
DRD5 P21918 2/20 0.31
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
AVPR1A P37288 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755760 1.00 PIK3CA (0.36) PIK3CACHRNB2CHRNA4YTHDC1LRRK2
SCHEMBL4755548 0.88 PDE4B (0.35) PIK3CALRRK2PDE1APDE1BPDE1C
SCHEMBL4755555 0.88 PDE4B (0.35) PIK3CALRRK2PDE1APDE1BPDE1C
SCHEMBL4755225 0.87 DRD1 (0.40) DRD1DRD5AVPR1A
SCHEMBL4755228 0.87 DRD1 (0.40) DRD1DRD5AVPR1A
SCHEMBL4756551 0.87 DRD1 (0.40) DRD1DRD5AVPR1A
SCHEMBL4755767 0.79 CHRNB2 (0.34) PIK3CACHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4755765 0.79 CHRNB2 (0.34) PIK3CACHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4755529 0.79 DRD1 (0.39) DRD1DRD5AVPR1A
SCHEMBL4755531 0.79 DRD1 (0.39) DRD1DRD5AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO claimed