SCHEMBL4756478

SCHEMBL4756478

Cc1cc(=O)n(-c2ccc(Cl)nc2)c(C2CC3C(C2)C3(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.36
CHRNA4 P43681 4/20 0.36
CYP11B2 P19099 1/20 0.34
CHRNB4 P30926 3/20 0.33
CHRNA3 P32297 3/20 0.33
PIK3CA P42336 2/20 0.32
USP14 P54578 1/20 0.32
POLB P06746 1/20 0.31
CRHR1 P34998 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985504 1.00 CHRNB2 (0.36) CHRNB2CHRNA4CYP11B2CHRNB4CHRNA3
SCHEMBL13985522 0.87 CRHR1 (0.41) POLBCRHR1
SCHEMBL4756481 0.87 CRHR1 (0.41) POLBCRHR1
SCHEMBL13985419 0.85 PDE4B (0.34) PIK3CAUSP14
SCHEMBL4755765 0.81 CHRNB2 (0.34) CHRNB2CHRNA4CHRNB4CHRNA3PIK3CA
SCHEMBL4755767 0.81 CHRNB2 (0.34) CHRNB2CHRNA4CHRNB4CHRNA3PIK3CA
SCHEMBL13660414 0.76 SMN1; SMN2 (0.34) CHRNB2CHRNA4CYP11B2POLB
SCHEMBL13660308 0.75 CHRNB2 (0.31) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL13660461 0.75 HRH3 (0.37) CHRNB2CHRNA4CYP11B2CHRNB4CHRNA3
SCHEMBL13985523 0.73 PIK3CA (0.37) CHRNB2CHRNA4CHRNB4CHRNA3PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed