SCHEMBL13660308

SCHEMBL13660308

O=c1c2ncsc2nc([C@H]2C[C@@H]3[C@H](C2)C3(F)F)n1-c1ccc(Cl)nc1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13660462 0.90 POLB (0.34)
SCHEMBL13660414 0.80 SMN1; SMN2 (0.34) CHRNB2CHRNA4
SCHEMBL13660461 0.80 HRH3 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL13985504 0.75 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL4756478 0.75 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL13660458 0.75 DRD1 (0.35)
SCHEMBL13660314 0.73 PDE4B (0.34)
SCHEMBL3169620 0.70 DRD1 (0.37)
SCHEMBL3169614 0.70 DRD1 (0.37)
SCHEMBL13660412 0.69 HRH3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009121036-A2 SUBSTITUTED ARYL PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2009-10-01 WO disclosed