SCHEMBL4756925

SCHEMBL4756925

CCOC(=O)c1cc(Cl)cc(C2CCN(CC(F)F)CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.41
CACNA1I Q9P0X4 3/20 0.41
FDFT1 P37268 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
ADAM17 P78536 2/20 0.39
HTR3E A5X5Y0 1/20 0.39
GMNN O75496 1/20 0.39
HTR3B O95264 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
MTOR P42345 1/20 0.39
HTR3A P46098 1/20 0.39
PMP22 Q01453 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755716 0.94 PDE4B (0.39) KCNH2CACNA1IFDFT1OPRM1OPRD1
SCHEMBL4755073 0.84 FDFT1 (0.39) FDFT1OPRM1OPRD1OPRK1ADAM17
SCHEMBL4758285 0.81 MAPT (0.43) FDFT1ADAM17TSHRHSD17B10GAA
SCHEMBL4757884 0.79 ALDH1A1 (0.54) ALOX15DPP4GAAMAPTALDH1A1
SCHEMBL4755037 0.77 CA12 (0.42) ALDH1A1MAPK1SMN1; SMN2NPSR1HPGD
SCHEMBL4756906 0.73 SLC6A2 (0.43) HTR3A
SCHEMBL17290064 0.70 SLC18A3 (0.46) TSHRHSD17B10GAASLC18A3ALDH1A1
SCHEMBL7589274 0.70 CA12 (0.62) CYP1A2CYP2D6NPSR1MEN1KMT2A
SCHEMBL2662880 0.70 CA12 (0.62) CYP1A2TSHRMEN1KMT2A
SCHEMBL4755119 0.70 PDE4A (0.45) TSHRGAAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed