SCHEMBL4755073

SCHEMBL4755073

CCOC(=O)c1cc(Cl)cc(C2CCN(CC(F)(F)F)CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
KDM1A O60341 1/20 0.37
ADAM17 P78536 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
RECQL P46063 1/20 0.36
CREBBP Q92793 1/20 0.36
HPGD P15428 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ALDH1A1 P00352 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756925 0.84 KCNH2 (0.41) FDFT1OPRM1OPRD1OPRK1ADAM17
SCHEMBL4755716 0.81 PDE4B (0.39) FDFT1OPRM1OPRD1OPRK1ADAM17
SCHEMBL4757884 0.79 ALDH1A1 (0.54) SMN1; SMN2NPSR1MEN1KMT2AHPGD
SCHEMBL4755037 0.77 CA12 (0.42) SMN1; SMN2NPSR1HPGDCA12CA1
SCHEMBL4758285 0.76 MAPT (0.43) FDFT1ADAM17SMN1; SMN2NPSR1MEN1
SCHEMBL4756934 0.73 PPARG (0.44) HPGDALDH1A1MAPTDRD2
SCHEMBL4756906 0.73 SLC6A2 (0.43) CA12CA1CA2CA7CA9
SCHEMBL16056333 0.70 FDFT1 (0.38) FDFT1NPSR1CA12CA1CA2
SCHEMBL25280227 0.70 HPGDS (0.45) KDM1ASMN1; SMN2HPGDALDH1A1
SCHEMBL7589274 0.70 CA12 (0.62) NPSR1MEN1KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed