SCHEMBL4756946

SCHEMBL4756946

Cc1cn(-c2cc(Cl)cc(C(=O)OCC(C)C)c2)c(C)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.42
PLA2G1B P04054 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
JMJD6 Q6NYC1 1/20 0.37
GRM5 P41594 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RECQL P46063 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
CACNA1F O60840 1/20 0.34
CACNA1D Q01668 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34
GABRA2 P47869 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756971 0.82 ALDH1A1 (0.41) GRM5ALDH1A1TSHRMEN1MAPT
SCHEMBL4757757 0.79 GPR119 (0.43) GRM5ALDH1A1TSHRCYP2C19NPSR1
SCHEMBL4757752 0.78 TPMT (0.47) GRM5ALDH1A1TSHRNPSR1MEN1
SCHEMBL5869072 0.70 ALOX15 (0.55) ALDH1A1MEN1KMT2AGABRA2GABRB2
SCHEMBL6580266 0.69 ALDH1A1 (0.59) GPR35PLA2G1BATG4BJMJD6ALDH1A1
SCHEMBL6057293 0.67 CHRM2 (0.55) GPR35JMJD6ALDH1A1TSHRCYP2C19
SCHEMBL6057138 0.65 ALDH1A1 (0.55) GPR35PLA2G1BATG4BALDH1A1TSHR
SCHEMBL9639553 0.65 ALDH1A1 (0.50) GPR35PLA2G1BATG4BJMJD6ALDH1A1
SCHEMBL559800 0.65 GPR35 (0.53) GPR35PLA2G1BATG4BJMJD6ALDH1A1
SCHEMBL20068189 0.64 ESR1 (0.58) GPR35PLA2G1BATG4BJMJD6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed