SCHEMBL4758202

SCHEMBL4758202

COc1ccc2nc(CCN3CCC(NC(=O)O)C(F)C3)c(=O)[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
EGFR P00533 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KCNH2 Q12809 4/20 0.40
EGLN1 Q9GZT9 1/20 0.40
JAK1 P23458 4/20 0.39
JAK2 O60674 3/20 0.39
TYK2 P29597 3/20 0.39
JAK3 P52333 3/20 0.39
FPR2 P25090 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TPH1 P17752 1/20 0.38
TPH2 Q8IWU9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4439862 0.91 POLB (0.43) POLBEGFRNPC1RAB9ASMN1; SMN2
SCHEMBL4441079 0.78 SMN1; SMN2 (0.42) POLBEGFRNPC1RAB9ASMN1; SMN2
SCHEMBL4733245 0.76 NPSR1 (0.46) EGFRNPC1RAB9ASMN1; SMN2EGLN1
SCHEMBL3357330 0.76 KCNH2 (0.66) KCNH2
SCHEMBL3838947 0.72 MPO (0.40) EGFRKCNH2
SCHEMBL5048771 0.71 KCNH2 (0.46) EGFRKCNH2TPH1TPH2
SCHEMBL5047886 0.71 SIGMAR1 (0.38) KCNH2
SCHEMBL5047682 0.70 CCR3 (0.41)
SCHEMBL16487837 0.69 CYP1A2 (0.51) POLBEGFRNPC1RAB9ASMN1; SMN2
SCHEMBL4444391 0.68 TP53 (0.40) SMN1; SMN2KCNH2KDM4EALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001126-A1 SUBSTITUTED PIPERIDINE DERIVATIVES AND THEIR USE AS ANTIBATERIAL AGENTS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed